Assay Detail

CHEMBL5474467

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Binding

Selectivity interaction (Inhibition of ex vivo anti-IgM/IL-4 -induced proximal pAKT formation in rats) EUB0000877a PIK3CD

ChEMBL ↗

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Target

Unchecked (CHEMBL612545) ↗

Open DB target context

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Unchecked (CHEMBL612545) is the working anchor for this assay review. Loading the live Open DB target snapshot…

Primary target Unchecked

CHEMBL612545

Anchored from Assay target.

Protein identity Unchecked

Disease frame Disease evidence pending

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Review focus Open DB context pending

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Total Activities

Compounds Tested

Activity Types

Assay Parameters

Assay Information

Assay Type	Binding
Category	Selectivity assay
Confidence	0 — Uncurated / Unknown
Curated By	Autocuration

Target

Unchecked (CHEMBL612545) ↗

Type

UNCHECKED

Publication

Selectivity Literature for EUbOPEN Chemogenomic Library

EUbOPEN
(2024)
· DOI

Activity Statistics

Type	Count	Avg pChEMBL	Best pChEMBL
EC50	1	7.08	7.08

Assay Parameters

Parameter	Type	Value	Units	Text
Protein family	Protein family	-	—	Protein kinase

Compounds Tested

Compound	Name	Phase	Activities	Best pChEMBL
CHEMBL3643413	LENIOLISIB	4.0	1	7.08

Activity Data

Compound	Name	Type	Rel.	Value	Units	pChEMBL
CHEMBL3643413	LENIOLISIB	EC50	=	83.0	nM	7.08