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Assay Detail

CHEMBL5474468

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Selectivity interaction (Rat whole blood B cell activation assay) EUB0000877a PIK3CD
1
Total Activities
1
Compounds Tested
1
Activity Types
1
Assay Parameters

Assay Information

Assay Type Binding
Tissue Blood
Category Selectivity assay
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Selectivity Literature for EUbOPEN Chemogenomic Library
EUbOPEN
(2024)
· DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 7.00 7.00

Assay Parameters

Parameter Type Value Units Text
Protein family Protein family - Protein kinase

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3643413 LENIOLISIB 4.0 1 7.00

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3643413 LENIOLISIB IC50 = 99.0 nM 7.00