Assay Detail

CHEMBL5477691

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Binding

Selectivity interaction (RapidFire MS assay (using full-length mouse protein MGAT2)) EUB0001079a MGAT2

ChEMBL ↗

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Target

Unchecked (CHEMBL612545) ↗

Open DB target context

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Unchecked (CHEMBL612545) is the working anchor for this assay review. Loading the live Open DB target snapshot…

Primary target Unchecked

CHEMBL612545

Anchored from Assay target.

Protein identity Unchecked

Disease frame Disease evidence pending

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Review focus Open DB context pending

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Total Activities

Compounds Tested

Activity Types

Assay Parameters

Assay Information

Assay Type	Binding
Category	Selectivity assay
Confidence	0 — Uncurated / Unknown
Curated By	Autocuration

Target

Unchecked (CHEMBL612545) ↗

Type

UNCHECKED

Publication

Selectivity Literature for EUbOPEN Chemogenomic Library

EUbOPEN
(2024)
· DOI

Activity Statistics

Type	Count	Avg pChEMBL	Best pChEMBL
IC50	1	6.28	6.28

Assay Parameters

Parameter	Type	Value	Units	Text
Protein family	Protein family	-	—	Transferase

Compounds Tested

Compound	Name	Phase	Activities	Best pChEMBL
CHEMBL4585920	TP-020n	—	1	6.28

Activity Data

Compound	Name	Type	Rel.	Value	Units	pChEMBL
CHEMBL4585920	TP-020n	IC50	=	530.0	nM	6.28