Assay Detail
Binding
CHEMBL5479529
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Selectivity interaction (Solid-phase-binding kinetics measurements (SPR using avi-tag biotinylated BUB1 catalytic domain)) EUB0001548a BUB1
1
Total Activities
1
Compounds Tested
1
Activity Types
1
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Category | Selectivity assay |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Mitotic checkpoint serine/threonine-protein kinase BUB1 (CHEMBL1772932) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Selectivity Literature for EUbOPEN Chemogenomic Library
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 1 | 8.68 | 8.68 |
Assay Parameters
| Parameter | Type | Value | Units | Text |
|---|---|---|---|---|
| Protein family | Protein family | - | — | Protein kinase |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5084426 | — | — | 1 | 8.68 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5084426 | — | Kd | = | 2.1 | nM | 8.68 |