Assay Detail
Binding
CHEMBL5505407
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of USP1 (unknown origin)
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Ubiquitin carboxyl-terminal hydrolase 1 (CHEMBL1795087) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
New Horizons of Synthetic Lethality in Cancer: Current Development and Future Perspectives.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 7.96 | 7.96 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5095186 | KSQ-4279 | — | 1 | 7.96 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5095186 | KSQ-4279 | IC50 | = | 11.0 | nM | 7.96 |