Assay Detail
Binding
CHEMBL5505418
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Agonist activity at PARG (unknown origin)
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
New Horizons of Synthetic Lethality in Cancer: Current Development and Future Perspectives.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 3 | 6.90 | 7.72 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4290954 | — | — | 1 | 7.72 |
| CHEMBL4286938 | — | — | 1 | 7.58 |
| CHEMBL4287730 | — | — | 1 | 5.41 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4290954 | — | EC50 | = | 19.0 | nM | 7.72 |
| CHEMBL4286938 | — | EC50 | = | 26.0 | nM | 7.58 |
| CHEMBL4287730 | — | EC50 | = | 3900.0 | nM | 5.41 |