Assay Detail
Binding
CHEMBL5505735
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of human recombinant Leucine aminopeptidase 3
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
ERAP Inhibitors in Autoimmunity and Immuno-Oncology: Medicinal Chemistry Insights.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 8.80 | 9.30 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL29292 | UBENIMEX | 2.0 | 1 | 9.30 |
| CHEMBL2103847 | TOSEDOSTAT | 2.0 | 1 | 8.30 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL29292 | UBENIMEX | IC50 | = | 0.5 | nM | 9.30 |
| CHEMBL2103847 | TOSEDOSTAT | IC50 | = | 5.0 | nM | 8.30 |