Assay Detail
Functional
CHEMBL5511081
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antiproliferative activity against human GL261 cells incubated for 72 hrs by MTT assay
29
Total Activities
29
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | GL261 |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Discovery of Novel Small-Molecule-Based Potential PD-L1/EGFR Dual Inhibitors with High Druggability for Glioblastoma Immunotherapy.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 29 | 5.52 | 5.92 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5559947 | — | — | 1 | 5.92 |
| CHEMBL5556281 | — | — | 1 | 5.91 |
| CHEMBL5564226 | — | — | 1 | 5.75 |
| CHEMBL5558740 | — | — | 1 | 5.71 |
| CHEMBL5555620 | — | — | 1 | 5.67 |
| CHEMBL5517715 | — | — | 1 | 5.65 |
| CHEMBL5523403 | — | — | 1 | 5.65 |
| CHEMBL5560649 | — | — | 1 | 5.62 |
| CHEMBL5560076 | — | — | 1 | 5.58 |
| CHEMBL5558842 | — | — | 1 | 5.57 |
| CHEMBL5562753 | — | — | 1 | 5.56 |
| CHEMBL5558630 | — | — | 1 | 5.49 |
| CHEMBL5562495 | — | — | 1 | 5.49 |
| CHEMBL5523580 | — | — | 1 | 5.48 |
| CHEMBL5565051 | — | — | 1 | 5.26 |
| CHEMBL4089730 | — | — | 1 | 5.24 |
| CHEMBL5559858 | — | — | 1 | 5.16 |
| CHEMBL939 | GEFITINIB | 4.0 | 1 | 4.67 |
| CHEMBL5556352 | — | — | 1 | - |
| CHEMBL5561232 | — | — | 1 | - |
| CHEMBL5557155 | — | — | 1 | - |
| CHEMBL5537075 | — | — | 1 | - |
| CHEMBL5532015 | — | — | 1 | - |
| CHEMBL5558514 | — | — | 1 | - |
| CHEMBL5555786 | — | — | 1 | - |
| CHEMBL5566977 | — | — | 1 | - |
| CHEMBL5556032 | — | — | 1 | - |
| CHEMBL4639202 | — | — | 1 | - |
| CHEMBL5562572 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5559947 | — | IC50 | = | 1190.0 | nM | 5.92 |
| CHEMBL5556281 | — | IC50 | = | 1240.0 | nM | 5.91 |
| CHEMBL5564226 | — | IC50 | = | 1790.0 | nM | 5.75 |
| CHEMBL5558740 | — | IC50 | = | 1970.0 | nM | 5.71 |
| CHEMBL5555620 | — | IC50 | = | 2160.0 | nM | 5.67 |
| CHEMBL5517715 | — | IC50 | = | 2250.0 | nM | 5.65 |
| CHEMBL5523403 | — | IC50 | = | 2240.0 | nM | 5.65 |
| CHEMBL5560649 | — | IC50 | = | 2390.0 | nM | 5.62 |
| CHEMBL5560076 | — | IC50 | = | 2630.0 | nM | 5.58 |
| CHEMBL5558842 | — | IC50 | = | 2720.0 | nM | 5.57 |
| CHEMBL5562753 | — | IC50 | = | 2760.0 | nM | 5.56 |
| CHEMBL5558630 | — | IC50 | = | 3220.0 | nM | 5.49 |
| CHEMBL5562495 | — | IC50 | = | 3250.0 | nM | 5.49 |
| CHEMBL5523580 | — | IC50 | = | 3300.0 | nM | 5.48 |
| CHEMBL5565051 | — | IC50 | = | 5460.0 | nM | 5.26 |
| CHEMBL4089730 | — | IC50 | = | 5720.0 | nM | 5.24 |
| CHEMBL5559858 | — | IC50 | = | 6860.0 | nM | 5.16 |
| CHEMBL939 | GEFITINIB | IC50 | = | 21540.0 | nM | 4.67 |
| CHEMBL5556352 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL5561232 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL5557155 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL5537075 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL5532015 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL5558514 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL5555786 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL5566977 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL5556032 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL4639202 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL5562572 | — | IC50 | > | 20000.0 | nM | - |