Assay Detail
Binding
CHEMBL5513517
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of MCT1 in human SiHa cells by lactate reporter assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | SiHa |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
pH regulators and their inhibitors in tumor microenvironment.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 6.65 | 7.23 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2442509 | — | — | 1 | 7.23 |
| CHEMBL1303766 | — | — | 1 | 6.07 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2442509 | — | IC50 | = | 59.0 | nM | 7.23 |
| CHEMBL1303766 | — | IC50 | = | 860.0 | nM | 6.07 |