Assay Detail
Binding
CHEMBL5513518
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Inhibition of MCT1 (unknown origin)
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
pH regulators and their inhibitors in tumor microenvironment.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 5.73 | 6.39 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL151 | LUTEOLIN | 2.0 | 1 | 6.39 |
| CHEMBL45068 | PHLORETIN | — | 1 | 5.59 |
| CHEMBL28626 | MORIN | — | 1 | 5.21 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL151 | LUTEOLIN | IC50 | = | 410.0 | nM | 6.39 |
| CHEMBL45068 | PHLORETIN | IC50 | = | 2570.0 | nM | 5.59 |
| CHEMBL28626 | MORIN | IC50 | = | 6210.0 | nM | 5.21 |