Assay Detail
Binding
CHEMBL5513546
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Inhibition of human CA IX by stopped flow CO2 hydrase assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
pH regulators and their inhibitors in tumor microenvironment.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 7.28 | 7.57 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5177984 | — | — | 1 | 7.57 |
| CHEMBL310671 | SACCHARIN | 3.0 | 1 | 6.99 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5177984 | — | Ki | = | 27.0 | nM | 7.57 |
| CHEMBL310671 | SACCHARIN | Ki | = | 103.0 | nM | 6.99 |