Assay Detail
Binding
CHEMBL5513555
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of human CA IX incubated for 15 to 4320 mins by by stopped-flow instrument based assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
pH regulators and their inhibitors in tumor microenvironment.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 6.72 | 6.72 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL12252 | 5,7-DIHYDROXY-4-METHYLCOUMARIN | — | 1 | 6.72 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL12252 | 5,7-DIHYDROXY-4-METHYLCOUMARIN | Ki | = | 190.0 | nM | 6.72 |