Assay Detail
Binding
CHEMBL5513615
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of His6-tagged Max (151 residues)(unknown origin) expressed in bacterial system/recombinant MYC ) (unknown origin) expressed in bacterial system by EMSA
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 7 — Homologous single protein target |
| Curated By | Autocuration |
Publication
MYC the oncogene from hell: Novel opportunities for cancer therapy.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 4.48 | 4.48 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1336889 | — | — | 1 | 4.48 |
| CHEMBL4286890 | — | — | 1 | 4.47 |
| CHEMBL2312756 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1336889 | — | IC50 | = | 33000.0 | nM | 4.48 |
| CHEMBL4286890 | — | IC50 | = | 34000.0 | nM | 4.47 |
| CHEMBL2312756 | — | IC50 | = | 146000.0 | nM | - |