Assay Detail
Functional
CHEMBL5513914
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antagonist activity at H1 receptor (unknown origin)
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Discovery of the novel and potent histamine H1 receptor antagonists for treatment of allergic diseases.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 9.08 | 9.08 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1172 | DESLORATADINE | 4.0 | 1 | 9.08 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1172 | DESLORATADINE | IC50 | = | 0.83 | nM | 9.08 |