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Assay Detail

CHEMBL5514817

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against SARS-CoV-2 infected in African green monkey Vero cells assessed as inhibition of viral replication pretreated with compound for 2 hr followed by viral infection and measured after 48 hrs by indirect immunofluorescence assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Severe acute respiratory syndrome coronavirus 2
Cell Type Vero
Confidence 1 — Organism
Curated By Autocuration

Target

SARS-CoV-2 (CHEMBL4303835)
Type ORGANISM
Organism Severe acute respiratory syndrome coronavirus 2

Publication

Structure-based discovery of potent myosin inhibitors to guide antiparasite drug development.
Tan X, Qu S, Wang G, Zhang G, Liu T, Ling F, Wang G.
Eur J Med Chem (2024) 269 : 116338 -116338
PubMed 38522112 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 1 8.10 8.10

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1201746 PRALATREXATE 4.0 1 8.10

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1201746 PRALATREXATE EC50 = 8.0 nM 8.10