Assay Detail
Binding
CHEMBL5522710
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Binding affinity to N-terminal His-tagged human recombinant RBP4 (19 to 201 residues) expressed in Escherichia coli BL21 (DE3) assessed as inhibition constant by ELISA method
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Recent Advances on Small-Molecule Inhibitors of Lipocalin-like Proteins.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 8.08 | 8.08 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL986 | RETINOL | 4.0 | 1 | 8.08 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL986 | RETINOL | Ki | = | 8.3 | nM | 8.08 |