Assay Detail
Binding
CHEMBL5524593
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Inhibition of SPTLC2 (unknown origin)
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Modulators for palmitoylation of proteins and small molecules.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 4 | 9.28 | 9.62 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5561881 | — | — | 1 | 9.62 |
| CHEMBL4228472 | — | — | 1 | 9.29 |
| CHEMBL4225519 | — | — | 1 | 9.12 |
| CHEMBL5565596 | — | — | 1 | 9.10 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5561881 | — | IC50 | = | 0.24 | nM | 9.62 |
| CHEMBL4228472 | — | IC50 | = | 0.51 | nM | 9.29 |
| CHEMBL4225519 | — | IC50 | = | 0.76 | nM | 9.12 |
| CHEMBL5565596 | — | IC50 | = | 0.8 | nM | 9.10 |