Assay Detail
Binding
CHEMBL5524640
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Inhibition of N-terminal His-tagged mouse GOAT expressed in baculovirus infected insect cells
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Mus musculus |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Modulators for palmitoylation of proteins and small molecules.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 4 | 5.47 | 6.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5556384 | — | — | 1 | 6.70 |
| CHEMBL5559872 | — | — | 1 | 5.16 |
| CHEMBL5542716 | — | — | 1 | 5.12 |
| CHEMBL5563229 | — | — | 1 | 4.88 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5556384 | — | IC50 | = | 200.0 | nM | 6.70 |
| CHEMBL5559872 | — | IC50 | = | 7000.0 | nM | 5.16 |
| CHEMBL5542716 | — | IC50 | = | 7540.0 | nM | 5.12 |
| CHEMBL5563229 | — | IC50 | = | 13100.0 | nM | 4.88 |