Assay Detail
Functional
CHEMBL5525277
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Antiproliferative activity against human U-266 cells incubated for 48 hrs by MTS assay
19
Total Activities
19
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | U-266 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Identification of novel GSPT1 degraders by virtual screening and bioassay.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 19 | 5.31 | 7.40 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4742712 | — | — | 1 | 7.40 |
| CHEMBL5566691 | — | — | 1 | 5.51 |
| CHEMBL5566579 | — | — | 1 | 5.42 |
| CHEMBL5561572 | — | — | 1 | 5.41 |
| CHEMBL5560999 | — | — | 1 | 5.17 |
| CHEMBL2000584 | — | — | 1 | 5.15 |
| CHEMBL5568165 | — | — | 1 | 4.99 |
| CHEMBL5542599 | — | — | 1 | 4.76 |
| CHEMBL5560535 | — | — | 1 | 4.75 |
| CHEMBL3208197 | — | — | 1 | 4.58 |
| CHEMBL5566890 | — | — | 1 | - |
| CHEMBL3214424 | — | — | 1 | - |
| CHEMBL5556820 | — | — | 1 | - |
| CHEMBL5555117 | — | — | 1 | - |
| CHEMBL5559758 | — | — | 1 | - |
| CHEMBL3195690 | — | — | 1 | - |
| CHEMBL5561994 | — | — | 1 | - |
| CHEMBL5562054 | — | — | 1 | - |
| CHEMBL5568413 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4742712 | — | IC50 | = | 40.0 | nM | 7.40 |
| CHEMBL5566691 | — | IC50 | = | 3100.0 | nM | 5.51 |
| CHEMBL5566579 | — | IC50 | = | 3800.0 | nM | 5.42 |
| CHEMBL5561572 | — | IC50 | = | 3930.0 | nM | 5.41 |
| CHEMBL5560999 | — | IC50 | = | 6750.0 | nM | 5.17 |
| CHEMBL2000584 | — | IC50 | = | 7130.0 | nM | 5.15 |
| CHEMBL5568165 | — | IC50 | = | 10140.0 | nM | 4.99 |
| CHEMBL5542599 | — | IC50 | = | 17450.0 | nM | 4.76 |
| CHEMBL5560535 | — | IC50 | = | 17670.0 | nM | 4.75 |
| CHEMBL3208197 | — | IC50 | = | 26590.0 | nM | 4.58 |
| CHEMBL5566890 | — | IC50 | > | 40000.0 | nM | - |
| CHEMBL3214424 | — | IC50 | > | 40000.0 | nM | - |
| CHEMBL5556820 | — | IC50 | > | 40000.0 | nM | - |
| CHEMBL5555117 | — | IC50 | > | 40000.0 | nM | - |
| CHEMBL5559758 | — | IC50 | > | 40000.0 | nM | - |
| CHEMBL3195690 | — | IC50 | > | 40000.0 | nM | - |
| CHEMBL5561994 | — | IC50 | > | 40000.0 | nM | - |
| CHEMBL5562054 | — | IC50 | > | 40000.0 | nM | - |
| CHEMBL5568413 | — | IC50 | > | 40000.0 | nM | - |