Assay Detail
Functional
CHEMBL5525280
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antiproliferative activity against human OCI-AML2 cells incubated for 48 hrs by MTS assay
19
Total Activities
19
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | OCI-AML2 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Identification of novel GSPT1 degraders by virtual screening and bioassay.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 19 | 5.49 | 8.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4742712 | — | — | 1 | 8.00 |
| CHEMBL5566691 | — | — | 1 | 5.60 |
| CHEMBL5566579 | — | — | 1 | 5.58 |
| CHEMBL5561572 | — | — | 1 | 5.58 |
| CHEMBL2000584 | — | — | 1 | 5.57 |
| CHEMBL5560999 | — | — | 1 | 5.05 |
| CHEMBL5542599 | — | — | 1 | 4.98 |
| CHEMBL5568165 | — | — | 1 | 4.96 |
| CHEMBL3208197 | — | — | 1 | 4.81 |
| CHEMBL5560535 | — | — | 1 | 4.77 |
| CHEMBL5566890 | — | — | 1 | - |
| CHEMBL3214424 | — | — | 1 | - |
| CHEMBL5556820 | — | — | 1 | - |
| CHEMBL5555117 | — | — | 1 | - |
| CHEMBL5559758 | — | — | 1 | - |
| CHEMBL3195690 | — | — | 1 | - |
| CHEMBL5561994 | — | — | 1 | - |
| CHEMBL5562054 | — | — | 1 | - |
| CHEMBL5568413 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4742712 | — | IC50 | = | 10.0 | nM | 8.00 |
| CHEMBL5566691 | — | IC50 | = | 2490.0 | nM | 5.60 |
| CHEMBL5566579 | — | IC50 | = | 2640.0 | nM | 5.58 |
| CHEMBL5561572 | — | IC50 | = | 2660.0 | nM | 5.58 |
| CHEMBL2000584 | — | IC50 | = | 2680.0 | nM | 5.57 |
| CHEMBL5560999 | — | IC50 | = | 8980.0 | nM | 5.05 |
| CHEMBL5542599 | — | IC50 | = | 10420.0 | nM | 4.98 |
| CHEMBL5568165 | — | IC50 | = | 11020.0 | nM | 4.96 |
| CHEMBL3208197 | — | IC50 | = | 15570.0 | nM | 4.81 |
| CHEMBL5560535 | — | IC50 | = | 17150.0 | nM | 4.77 |
| CHEMBL5566890 | — | IC50 | > | 40000.0 | nM | - |
| CHEMBL3214424 | — | IC50 | > | 40000.0 | nM | - |
| CHEMBL5556820 | — | IC50 | > | 40000.0 | nM | - |
| CHEMBL5555117 | — | IC50 | > | 40000.0 | nM | - |
| CHEMBL5559758 | — | IC50 | > | 40000.0 | nM | - |
| CHEMBL3195690 | — | IC50 | > | 40000.0 | nM | - |
| CHEMBL5561994 | — | IC50 | > | 40000.0 | nM | - |
| CHEMBL5562054 | — | IC50 | > | 40000.0 | nM | - |
| CHEMBL5568413 | — | IC50 | > | 40000.0 | nM | - |