Assay Detail
Binding
CHEMBL5527155
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of MAO-A (unknown origin) measured by MAO-GloTM method
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Natural Product-Inspired Dopamine Receptor Ligands.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 4.56 | 5.07 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL151 | LUTEOLIN | 2.0 | 1 | 5.07 |
| CHEMBL228430 | — | — | 1 | 4.05 |
| CHEMBL470234 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL151 | LUTEOLIN | IC50 | = | 8570.0 | nM | 5.07 |
| CHEMBL228430 | — | IC50 | = | 89310.0 | nM | 4.05 |
| CHEMBL470234 | — | IC50 | = | 204940.0 | nM | - |