Assay Detail
Functional
CHEMBL5534280
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Agonist activity at human GCGR expressed in HEK293 cells assessed as cAMP level measured after 60 mins by HTRF based assay
28
Total Activities
28
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HEK293 |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Discovery of a Novel Glucagon-like Peptide-1 (GLP-1) Analogue from Bullfrog and Investigation of Its Potential for Designing GLP-1-Based Multiagonists.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 28 | 9.24 | 10.57 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5573719 | — | — | 1 | 10.57 |
| CHEMBL5573706 | — | — | 1 | 10.28 |
| CHEMBL5314341 | GLUCAGON | 4.0 | 1 | 10.04 |
| CHEMBL5575146 | — | — | 1 | 9.89 |
| CHEMBL5584018 | — | — | 1 | 9.82 |
| CHEMBL4297630 | COTADUTIDE | 2.0 | 1 | 9.77 |
| CHEMBL5584095 | — | — | 1 | 9.74 |
| CHEMBL5572101 | — | — | 1 | 9.72 |
| CHEMBL5590721 | — | — | 1 | 9.64 |
| CHEMBL5575497 | — | — | 1 | 9.29 |
| CHEMBL5579680 | — | — | 1 | 9.28 |
| CHEMBL5573864 | — | — | 1 | 9.28 |
| CHEMBL5570478 | — | — | 1 | 9.21 |
| CHEMBL5563008 | — | — | 1 | 9.21 |
| CHEMBL5574566 | — | — | 1 | 9.18 |
| CHEMBL5593907 | — | — | 1 | 9.10 |
| CHEMBL5571917 | — | — | 1 | 9.07 |
| CHEMBL5572113 | — | — | 1 | 9.04 |
| CHEMBL5590909 | — | — | 1 | 8.92 |
| CHEMBL5594986 | — | — | 1 | 8.85 |
| CHEMBL5569213 | — | — | 1 | 8.74 |
| CHEMBL5575699 | — | — | 1 | 8.74 |
| CHEMBL5570630 | — | — | 1 | 8.74 |
| CHEMBL5570738 | — | — | 1 | 8.59 |
| CHEMBL5571645 | — | — | 1 | 8.59 |
| CHEMBL5575723 | — | — | 1 | 8.51 |
| CHEMBL5565062 | — | — | 1 | 8.51 |
| CHEMBL5570925 | — | — | 1 | 8.46 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5573719 | — | EC50 | = | 0.027 | nM | 10.57 |
| CHEMBL5573706 | — | EC50 | = | 0.052 | nM | 10.28 |
| CHEMBL5314341 | GLUCAGON | EC50 | = | 0.092 | nM | 10.04 |
| CHEMBL5575146 | — | EC50 | = | 0.13 | nM | 9.89 |
| CHEMBL5584018 | — | EC50 | = | 0.15 | nM | 9.82 |
| CHEMBL4297630 | COTADUTIDE | EC50 | = | 0.17 | nM | 9.77 |
| CHEMBL5584095 | — | EC50 | = | 0.18 | nM | 9.74 |
| CHEMBL5572101 | — | EC50 | = | 0.19 | nM | 9.72 |
| CHEMBL5590721 | — | EC50 | = | 0.23 | nM | 9.64 |
| CHEMBL5575497 | — | EC50 | = | 0.51 | nM | 9.29 |
| CHEMBL5579680 | — | EC50 | = | 0.53 | nM | 9.28 |
| CHEMBL5573864 | — | EC50 | = | 0.53 | nM | 9.28 |
| CHEMBL5570478 | — | EC50 | = | 0.62 | nM | 9.21 |
| CHEMBL5563008 | — | EC50 | = | 0.61 | nM | 9.21 |
| CHEMBL5574566 | — | EC50 | = | 0.66 | nM | 9.18 |
| CHEMBL5593907 | — | EC50 | = | 0.8 | nM | 9.10 |
| CHEMBL5571917 | — | EC50 | = | 0.85 | nM | 9.07 |
| CHEMBL5572113 | — | EC50 | = | 0.91 | nM | 9.04 |
| CHEMBL5590909 | — | EC50 | = | 1.2 | nM | 8.92 |
| CHEMBL5594986 | — | EC50 | = | 1.4 | nM | 8.85 |
| CHEMBL5569213 | — | EC50 | = | 1.8 | nM | 8.74 |
| CHEMBL5575699 | — | EC50 | = | 1.8 | nM | 8.74 |
| CHEMBL5570630 | — | EC50 | = | 1.8 | nM | 8.74 |
| CHEMBL5570738 | — | EC50 | = | 2.6 | nM | 8.59 |
| CHEMBL5571645 | — | EC50 | = | 2.6 | nM | 8.59 |
| CHEMBL5575723 | — | EC50 | = | 3.1 | nM | 8.51 |
| CHEMBL5565062 | — | EC50 | = | 3.1 | nM | 8.51 |
| CHEMBL5570925 | — | EC50 | = | 3.5 | nM | 8.46 |