Assay Detail
Binding
CHEMBL5535210
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Inhibition of PI3K (unknown origin)
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Comprehensive Insights that Targeting PIM for Cancer Therapy: Prospects and Obstacles.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 8.84 | 9.89 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4878958 | — | — | 1 | 9.89 |
| CHEMBL4869696 | — | — | 1 | 7.78 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4878958 | — | IC50 | = | 0.13 | nM | 9.89 |
| CHEMBL4869696 | — | IC50 | = | 16.8 | nM | 7.78 |