Assay Detail
Functional
CHEMBL5536200
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antiproliferative activity against human Cisplatin and radiotherapy resistant CAL27RR cells incubated for 48 hrs by XTT assay
32
Total Activities
32
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | Cisplatin and radiotherapy resistant CAL27RR |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
A Potent Solution for Tumor Growth and Angiogenesis Suppression via an ELR<sup>+</sup>CXCL-CXCR1/2 Pathway Inhibitor.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 32 | 5.16 | 5.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5549970 | — | — | 1 | 5.70 |
| CHEMBL5579669 | — | — | 1 | 5.60 |
| CHEMBL5570017 | — | — | 1 | 5.60 |
| CHEMBL5568805 | — | — | 1 | 5.60 |
| CHEMBL4799715 | — | — | 1 | 5.40 |
| CHEMBL4550904 | — | — | 1 | 5.40 |
| CHEMBL5572121 | — | — | 1 | 5.40 |
| CHEMBL5570076 | — | — | 1 | 5.40 |
| CHEMBL5572632 | — | — | 1 | 5.22 |
| CHEMBL5565327 | — | — | 1 | 5.16 |
| CHEMBL5570451 | — | — | 1 | 5.16 |
| CHEMBL5583611 | — | — | 1 | 5.00 |
| CHEMBL5564096 | — | — | 1 | 4.82 |
| CHEMBL5594187 | — | — | 1 | 4.70 |
| CHEMBL5575595 | — | — | 1 | 4.70 |
| CHEMBL5573045 | — | — | 1 | 4.70 |
| CHEMBL5568724 | — | — | 1 | 4.70 |
| CHEMBL5568819 | — | — | 1 | 4.60 |
| CHEMBL5590695 | — | — | 1 | - |
| CHEMBL5567361 | — | — | 1 | - |
| CHEMBL5573468 | — | — | 1 | - |
| CHEMBL5563240 | — | — | 1 | - |
| CHEMBL5572383 | — | — | 1 | - |
| CHEMBL5555259 | — | — | 1 | - |
| CHEMBL5575771 | — | — | 1 | - |
| CHEMBL5594473 | — | — | 1 | - |
| CHEMBL5573651 | — | — | 1 | - |
| CHEMBL5571576 | — | — | 1 | - |
| CHEMBL5570892 | — | — | 1 | - |
| CHEMBL5572155 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5549970 | — | IC50 | = | 2000.0 | nM | 5.70 |
| CHEMBL5579669 | — | IC50 | = | 2500.0 | nM | 5.60 |
| CHEMBL5570017 | — | IC50 | = | 2500.0 | nM | 5.60 |
| CHEMBL5568805 | — | IC50 | = | 2500.0 | nM | 5.60 |
| CHEMBL4799715 | — | IC50 | = | 4000.0 | nM | 5.40 |
| CHEMBL4550904 | — | IC50 | = | 4000.0 | nM | 5.40 |
| CHEMBL5572121 | — | IC50 | = | 4000.0 | nM | 5.40 |
| CHEMBL5570076 | — | IC50 | = | 4000.0 | nM | 5.40 |
| CHEMBL5572632 | — | IC50 | = | 6000.0 | nM | 5.22 |
| CHEMBL5565327 | — | IC50 | = | 7000.0 | nM | 5.16 |
| CHEMBL5570451 | — | IC50 | = | 7000.0 | nM | 5.16 |
| CHEMBL5583611 | — | IC50 | = | 10000.0 | nM | 5.00 |
| CHEMBL5564096 | — | IC50 | = | 15000.0 | nM | 4.82 |
| CHEMBL5575595 | — | IC50 | = | 20000.0 | nM | 4.70 |
| CHEMBL5594187 | — | IC50 | = | 20000.0 | nM | 4.70 |
| CHEMBL5568724 | — | IC50 | = | 20000.0 | nM | 4.70 |
| CHEMBL5573045 | — | IC50 | = | 20000.0 | nM | 4.70 |
| CHEMBL5568819 | — | IC50 | = | 25000.0 | nM | 4.60 |
| CHEMBL5591275 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL5593327 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL5572155 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL5570892 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL5571576 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL5573651 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL5594473 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL5575771 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL5555259 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL5572383 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL5563240 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL5573468 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL5567361 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL5590695 | — | IC50 | > | 25000.0 | nM | - |