Assay Detail
Functional
CHEMBL5536201
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antiproliferative activity against human CAL-27 cells incubated for 48 hrs by XTT assay
32
Total Activities
32
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | CAL-27 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
A Potent Solution for Tumor Growth and Angiogenesis Suppression via an ELR<sup>+</sup>CXCL-CXCR1/2 Pathway Inhibitor.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 32 | 5.19 | 6.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5579669 | — | — | 1 | 6.00 |
| CHEMBL5568805 | — | — | 1 | 5.60 |
| CHEMBL5549970 | — | — | 1 | 5.52 |
| CHEMBL5572121 | — | — | 1 | 5.40 |
| CHEMBL4799715 | — | — | 1 | 5.30 |
| CHEMBL5570017 | — | — | 1 | 5.30 |
| CHEMBL5572632 | — | — | 1 | 5.16 |
| CHEMBL5570076 | — | — | 1 | 5.16 |
| CHEMBL5572383 | — | — | 1 | 5.16 |
| CHEMBL5565327 | — | — | 1 | 5.10 |
| CHEMBL5583611 | — | — | 1 | 4.60 |
| CHEMBL4550904 | — | — | 1 | 4.60 |
| CHEMBL5568724 | — | — | 1 | 4.60 |
| CHEMBL5593327 | — | — | 1 | - |
| CHEMBL5575595 | — | — | 1 | - |
| CHEMBL5564096 | — | — | 1 | - |
| CHEMBL5594187 | — | — | 1 | - |
| CHEMBL5572155 | — | — | 1 | - |
| CHEMBL5570451 | — | — | 1 | - |
| CHEMBL5570892 | — | — | 1 | - |
| CHEMBL5567361 | — | — | 1 | - |
| CHEMBL5573651 | — | — | 1 | - |
| CHEMBL5594473 | — | — | 1 | - |
| CHEMBL5575771 | — | — | 1 | - |
| CHEMBL5555259 | — | — | 1 | - |
| CHEMBL5563240 | — | — | 1 | - |
| CHEMBL5568819 | — | — | 1 | - |
| CHEMBL5573468 | — | — | 1 | - |
| CHEMBL5590695 | — | — | 1 | - |
| CHEMBL5571576 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5579669 | — | IC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL5568805 | — | IC50 | = | 2500.0 | nM | 5.60 |
| CHEMBL5549970 | — | IC50 | = | 3000.0 | nM | 5.52 |
| CHEMBL5572121 | — | IC50 | = | 4000.0 | nM | 5.40 |
| CHEMBL4799715 | — | IC50 | = | 5000.0 | nM | 5.30 |
| CHEMBL5570017 | — | IC50 | = | 5000.0 | nM | 5.30 |
| CHEMBL5572632 | — | IC50 | = | 7000.0 | nM | 5.16 |
| CHEMBL5570076 | — | IC50 | = | 7000.0 | nM | 5.16 |
| CHEMBL5572383 | — | IC50 | = | 7000.0 | nM | 5.16 |
| CHEMBL5565327 | — | IC50 | = | 8000.0 | nM | 5.10 |
| CHEMBL5568724 | — | IC50 | = | 25000.0 | nM | 4.60 |
| CHEMBL4550904 | — | IC50 | = | 25000.0 | nM | 4.60 |
| CHEMBL5583611 | — | IC50 | = | 25000.0 | nM | 4.60 |
| CHEMBL5573045 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL5591275 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL5593327 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL5575595 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL5564096 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL5594187 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL5572155 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL5570451 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL5570892 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL5567361 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL5573651 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL5594473 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL5575771 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL5555259 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL5563240 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL5568819 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL5573468 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL5590695 | — | IC50 | > | 25000.0 | nM | - |
| CHEMBL5571576 | — | IC50 | > | 25000.0 | nM | - |