Assay Detail
Binding
CHEMBL5536535
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Inhibition of STK17A (unknown origin) in presence of ATP
19
Total Activities
19
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Potent, Selective, and Orally Bioavailable Quinazoline-Based STK17A/B Dual Inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 19 | 7.47 | 7.92 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5573038 | — | — | 1 | 7.92 |
| CHEMBL5579785 | — | — | 1 | 7.77 |
| CHEMBL5574990 | — | — | 1 | 7.75 |
| CHEMBL5564156 | — | — | 1 | 7.72 |
| CHEMBL5569603 | — | — | 1 | 7.70 |
| CHEMBL5571334 | — | — | 1 | 7.70 |
| CHEMBL5569176 | — | — | 1 | 7.70 |
| CHEMBL5575519 | — | — | 1 | 7.68 |
| CHEMBL5575113 | — | — | 1 | 7.64 |
| CHEMBL5589781 | — | — | 1 | 7.60 |
| CHEMBL5573207 | — | — | 1 | 7.54 |
| CHEMBL5574107 | — | — | 1 | 7.37 |
| CHEMBL5565459 | — | — | 1 | 7.32 |
| CHEMBL5570123 | — | — | 1 | 7.29 |
| CHEMBL5542886 | — | — | 1 | 7.26 |
| CHEMBL5570883 | — | — | 1 | 7.18 |
| CHEMBL5571678 | — | — | 1 | 6.84 |
| CHEMBL5570247 | — | — | 1 | 6.50 |
| CHEMBL5569006 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5573038 | — | IC50 | = | 12.0 | nM | 7.92 |
| CHEMBL5579785 | — | IC50 | = | 17.0 | nM | 7.77 |
| CHEMBL5574990 | — | IC50 | = | 18.0 | nM | 7.75 |
| CHEMBL5564156 | — | IC50 | = | 19.0 | nM | 7.72 |
| CHEMBL5569603 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL5571334 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL5569176 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL5575519 | — | IC50 | = | 21.0 | nM | 7.68 |
| CHEMBL5575113 | — | IC50 | = | 23.0 | nM | 7.64 |
| CHEMBL5589781 | — | IC50 | = | 25.0 | nM | 7.60 |
| CHEMBL5573207 | — | IC50 | = | 29.0 | nM | 7.54 |
| CHEMBL5574107 | — | IC50 | = | 43.0 | nM | 7.37 |
| CHEMBL5565459 | — | IC50 | = | 48.0 | nM | 7.32 |
| CHEMBL5570123 | — | IC50 | = | 51.0 | nM | 7.29 |
| CHEMBL5542886 | — | IC50 | = | 55.0 | nM | 7.26 |
| CHEMBL5570883 | — | IC50 | = | 66.0 | nM | 7.18 |
| CHEMBL5571678 | — | IC50 | = | 144.0 | nM | 6.84 |
| CHEMBL5570247 | — | IC50 | = | 316.0 | nM | 6.50 |
| CHEMBL5569006 | — | IC50 | > | 10000.0 | nM | - |