Assay Detail
Binding
CHEMBL5538583
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of PARP7 (unknown origin) measured after 1 hr incubation by microplate reader assay
19
Total Activities
19
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Protein mono-ADP-ribosyltransferase TIPARP (CHEMBL2380188) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Discovery of Highly Selective PARP7 Inhibitors with a Novel Scaffold for Cancer Immunotherapy.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 19 | 7.58 | 8.35 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5571636 | — | — | 1 | 8.35 |
| CHEMBL5095043 | ATAMPARIB | 1.0 | 1 | 8.25 |
| CHEMBL5573525 | — | — | 1 | 8.07 |
| CHEMBL5570155 | — | — | 1 | 7.70 |
| CHEMBL5563046 | — | — | 1 | 7.65 |
| CHEMBL5571907 | — | — | 1 | 7.34 |
| CHEMBL5566904 | — | — | 1 | 7.21 |
| CHEMBL5572349 | — | — | 1 | 6.91 |
| CHEMBL5591356 | — | — | 1 | 6.77 |
| CHEMBL5569932 | — | — | 1 | - |
| CHEMBL5566250 | — | — | 1 | - |
| CHEMBL5564068 | — | — | 1 | - |
| CHEMBL5590832 | — | — | 1 | - |
| CHEMBL5562672 | — | — | 1 | - |
| CHEMBL5575757 | — | — | 1 | - |
| CHEMBL5572531 | — | — | 1 | - |
| CHEMBL5592601 | — | — | 1 | - |
| CHEMBL5567004 | — | — | 1 | - |
| CHEMBL5592002 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5571636 | — | IC50 | = | 4.5 | nM | 8.35 |
| CHEMBL5095043 | ATAMPARIB | IC50 | = | 5.6 | nM | 8.25 |
| CHEMBL5573525 | — | IC50 | = | 8.5 | nM | 8.07 |
| CHEMBL5570155 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL5563046 | — | IC50 | = | 22.3 | nM | 7.65 |
| CHEMBL5571907 | — | IC50 | = | 46.0 | nM | 7.34 |
| CHEMBL5566904 | — | IC50 | = | 62.0 | nM | 7.21 |
| CHEMBL5572349 | — | IC50 | = | 122.0 | nM | 6.91 |
| CHEMBL5591356 | — | IC50 | = | 171.3 | nM | 6.77 |
| CHEMBL5569932 | — | IC50 | - | — | - | |
| CHEMBL5566250 | — | IC50 | - | — | - | |
| CHEMBL5564068 | — | IC50 | - | — | - | |
| CHEMBL5590832 | — | IC50 | - | — | - | |
| CHEMBL5562672 | — | IC50 | - | — | - | |
| CHEMBL5575757 | — | IC50 | - | — | - | |
| CHEMBL5572531 | — | IC50 | - | — | - | |
| CHEMBL5592601 | — | IC50 | - | — | - | |
| CHEMBL5567004 | — | IC50 | - | — | - | |
| CHEMBL5592002 | — | IC50 | - | — | - |