Assay Detail
Functional
CHEMBL5539301
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antiproliferative activity against human MV4-11 cells harboring MLL-r assessed as cell growth inhibition incubated for 5 days by CCK-8 assay
15
Total Activities
14
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | MV4-11 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Discovery and Optimization of WDR5 Inhibitors via Cascade Deoxyribonucleic Acid-Encoded Library Selection Approach.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 15 | 5.47 | 6.77 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4588661 | — | — | 1 | 6.77 |
| CHEMBL5579746 | — | — | 1 | 5.72 |
| CHEMBL5572530 | — | — | 1 | 5.64 |
| CHEMBL5595245 | — | — | 1 | 5.47 |
| CHEMBL5579685 | — | — | 1 | 5.46 |
| CHEMBL5573553 | — | — | 1 | 5.41 |
| CHEMBL5574810 | — | — | 1 | 5.41 |
| CHEMBL5573350 | — | — | 2 | 5.38 |
| CHEMBL5592145 | — | — | 1 | 5.32 |
| CHEMBL5591718 | — | — | 1 | 5.32 |
| CHEMBL5562523 | — | — | 1 | 5.30 |
| CHEMBL5574474 | — | — | 1 | 5.26 |
| CHEMBL5572054 | — | — | 1 | 5.24 |
| CHEMBL5565914 | — | — | 1 | 5.21 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4588661 | — | IC50 | = | 170.0 | nM | 6.77 |
| CHEMBL5579746 | — | IC50 | = | 1900.0 | nM | 5.72 |
| CHEMBL5572530 | — | IC50 | = | 2300.0 | nM | 5.64 |
| CHEMBL5595245 | — | IC50 | = | 3400.0 | nM | 5.47 |
| CHEMBL5579685 | — | IC50 | = | 3500.0 | nM | 5.46 |
| CHEMBL5573553 | — | IC50 | = | 3900.0 | nM | 5.41 |
| CHEMBL5574810 | — | IC50 | = | 3930.0 | nM | 5.41 |
| CHEMBL5573350 | — | IC50 | = | 4130.0 | nM | 5.38 |
| CHEMBL5592145 | — | IC50 | = | 4800.0 | nM | 5.32 |
| CHEMBL5591718 | — | IC50 | = | 4800.0 | nM | 5.32 |
| CHEMBL5562523 | — | IC50 | = | 5000.0 | nM | 5.30 |
| CHEMBL5574474 | — | IC50 | = | 5500.0 | nM | 5.26 |
| CHEMBL5572054 | — | IC50 | = | 5700.0 | nM | 5.24 |
| CHEMBL5573350 | — | IC50 | = | 6200.0 | nM | 5.21 |
| CHEMBL5565914 | — | IC50 | = | 6200.0 | nM | 5.21 |