Assay Detail
Functional
CHEMBL5539302
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Antiproliferative activity against human K562 cells assessed as cell growth inhibition incubated for 5 days by CCK-8 assay
15
Total Activities
14
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | K562 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Discovery and Optimization of WDR5 Inhibitors via Cascade Deoxyribonucleic Acid-Encoded Library Selection Approach.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 15 | 5.39 | 5.96 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5579746 | — | — | 1 | 5.96 |
| CHEMBL5573553 | — | — | 1 | 5.52 |
| CHEMBL5574810 | — | — | 1 | 5.52 |
| CHEMBL5565914 | — | — | 1 | 5.47 |
| CHEMBL5573350 | — | — | 2 | 5.46 |
| CHEMBL5572530 | — | — | 1 | 5.46 |
| CHEMBL4588661 | — | — | 1 | 5.44 |
| CHEMBL5579685 | — | — | 1 | 5.40 |
| CHEMBL5592145 | — | — | 1 | 5.33 |
| CHEMBL5574474 | — | — | 1 | 5.31 |
| CHEMBL5595245 | — | — | 1 | 5.31 |
| CHEMBL5591718 | — | — | 1 | 5.28 |
| CHEMBL5572054 | — | — | 1 | 5.15 |
| CHEMBL5562523 | — | — | 1 | 4.91 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5579746 | — | IC50 | = | 1100.0 | nM | 5.96 |
| CHEMBL5573553 | — | IC50 | = | 3000.0 | nM | 5.52 |
| CHEMBL5574810 | — | IC50 | = | 3030.0 | nM | 5.52 |
| CHEMBL5565914 | — | IC50 | = | 3400.0 | nM | 5.47 |
| CHEMBL5573350 | — | IC50 | = | 3430.0 | nM | 5.46 |
| CHEMBL5572530 | — | IC50 | = | 3500.0 | nM | 5.46 |
| CHEMBL4588661 | — | IC50 | = | 3600.0 | nM | 5.44 |
| CHEMBL5579685 | — | IC50 | = | 4000.0 | nM | 5.40 |
| CHEMBL5592145 | — | IC50 | = | 4700.0 | nM | 5.33 |
| CHEMBL5574474 | — | IC50 | = | 4900.0 | nM | 5.31 |
| CHEMBL5573350 | — | IC50 | = | 4900.0 | nM | 5.31 |
| CHEMBL5595245 | — | IC50 | = | 4900.0 | nM | 5.31 |
| CHEMBL5591718 | — | IC50 | = | 5200.0 | nM | 5.28 |
| CHEMBL5572054 | — | IC50 | = | 7100.0 | nM | 5.15 |
| CHEMBL5562523 | — | IC50 | = | 12200.0 | nM | 4.91 |