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Assay Detail

CHEMBL5539895

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against SARS-CoV-2 infected in human Huh-7 cells assessed as reduction in viral growth
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Severe acute respiratory syndrome coronavirus 2
Confidence 1 — Organism
Curated By Autocuration

Target

SARS-CoV-2 (CHEMBL4303835)
Type ORGANISM
Organism Severe acute respiratory syndrome coronavirus 2

Publication

Hepatitis C: The Story of a Long Journey through First, Second, and Third Generation NS3/4A Peptidomimetic Inhibitors. What Did We Learn?
Martino SD, Petri GL, De Rosa M.
J Med Chem (2024) 67 : 885 -921
PubMed 38179950 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 4 7.76 8.40

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL414993 1 8.40
CHEMBL3125106 1 7.72
CHEMBL1956820 GS-9256 2.0 1 7.70
CHEMBL3128331 1 7.22

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL414993 EC50 = 4.0 nM 8.40
CHEMBL3125106 EC50 = 19.0 nM 7.72
CHEMBL1956820 GS-9256 EC50 = 20.0 nM 7.70
CHEMBL3128331 EC50 = 60.0 nM 7.22