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Assay Detail

CHEMBL5543313

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Anti-inflammatory activity against mouse J774.A1 cells assessed as inhibition of LPS-induced IL-1beta mRNA expression level pretreated for 30 mins followed by LPS-induction and measured after 6 hrs by RT-PCR analysis
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Mus musculus
Cell Type J774.A1
Confidence 1 — Organism
Curated By Autocuration

Target

J774.A1 (CHEMBL614040)
Type CELL-LINE
Organism Mus musculus

Publication

Discovery of anti-inflammatory natural flavonoids: Diverse scaffolds and promising leads for drug discovery.
Li J, Zhao R, Miao P, Xu F, Chen J, Jiang X, Hui Z, Wang L, Bai R.
Eur J Med Chem (2023) 260 : 115791 -115791
PubMed 37683361 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 4.37 4.37

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL317221 1 4.37

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL317221 IC50 = 42760.0 nM 4.37