Assay Detail
Functional
CHEMBL5546302
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Cytotoxicity against human HPAC cells assessed as inhibition of cell growth incubated for 72 hrs by MTT assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HPAC |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Lead Compound Development of SRC-3 Inhibitors with Improved Pharmacokinetic Properties and Anticancer Efficacy.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 7.58 | 7.58 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5590309 | — | — | 1 | 7.58 |
| CHEMBL5570209 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5590309 | — | IC50 | = | 26.0 | nM | 7.58 |
| CHEMBL5570209 | — | IC50 | - | — | - |