Assay Detail
Binding
CHEMBL5546604
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Inhibition of CDK2/CYCA (unknown origin)
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Recent Discovery and Development of Inhibitors that Target CDK9 and Their Therapeutic Indications.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 6.29 | 7.33 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5563573 | — | — | 1 | 7.33 |
| CHEMBL5287796 | — | — | 1 | 5.93 |
| CHEMBL3263773 | — | — | 1 | 5.61 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5563573 | — | IC50 | = | 47.0 | nM | 7.33 |
| CHEMBL5287796 | — | IC50 | = | 1180.0 | nM | 5.93 |
| CHEMBL3263773 | — | IC50 | = | 2441.0 | nM | 5.61 |