Assay Detail
Functional
CHEMBL5551971
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Cytotoxicity against human U-937 cells incubated for 24 hrs by CCK8 assay
11
Total Activities
11
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | U-937 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Synthesis and structural optimization of oncolytic peptide LTX-315.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 11 | 4.86 | 5.13 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5555708 | — | — | 1 | 5.13 |
| CHEMBL5570934 | — | — | 1 | 5.10 |
| CHEMBL4297628 | RUXOTEMITIDE | 2.0 | 1 | 4.97 |
| CHEMBL5570540 | — | — | 1 | 4.96 |
| CHEMBL5569031 | — | — | 1 | 4.91 |
| CHEMBL5572304 | — | — | 1 | 4.89 |
| CHEMBL5573214 | — | — | 1 | 4.87 |
| CHEMBL5569116 | — | — | 1 | 4.86 |
| CHEMBL5592571 | — | — | 1 | 4.51 |
| CHEMBL5574505 | — | — | 1 | 4.39 |
| CHEMBL5566343 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5555708 | — | IC50 | = | 7400.0 | nM | 5.13 |
| CHEMBL5570934 | — | IC50 | = | 8000.0 | nM | 5.10 |
| CHEMBL4297628 | RUXOTEMITIDE | IC50 | = | 10700.0 | nM | 4.97 |
| CHEMBL5570540 | — | IC50 | = | 11000.0 | nM | 4.96 |
| CHEMBL5569031 | — | IC50 | = | 12300.0 | nM | 4.91 |
| CHEMBL5572304 | — | IC50 | = | 12800.0 | nM | 4.89 |
| CHEMBL5573214 | — | IC50 | = | 13600.0 | nM | 4.87 |
| CHEMBL5569116 | — | IC50 | = | 13800.0 | nM | 4.86 |
| CHEMBL5592571 | — | IC50 | = | 31100.0 | nM | 4.51 |
| CHEMBL5574505 | — | IC50 | = | 40900.0 | nM | 4.39 |
| CHEMBL5566343 | — | IC50 | = | 203800.0 | nM | - |