Assay Detail
Functional
CHEMBL5551972
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Cytotoxicity against human CoC1 cells incubated for 24 hrs by CCK8 assay
11
Total Activities
11
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | CoC1 |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Synthesis and structural optimization of oncolytic peptide LTX-315.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 11 | 4.80 | 5.10 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5570934 | — | — | 1 | 5.10 |
| CHEMBL5555708 | — | — | 1 | 5.08 |
| CHEMBL5572304 | — | — | 1 | 4.93 |
| CHEMBL5570540 | — | — | 1 | 4.87 |
| CHEMBL5573214 | — | — | 1 | 4.85 |
| CHEMBL5569031 | — | — | 1 | 4.82 |
| CHEMBL4297628 | RUXOTEMITIDE | 2.0 | 1 | 4.78 |
| CHEMBL5569116 | — | — | 1 | 4.72 |
| CHEMBL5592571 | — | — | 1 | 4.44 |
| CHEMBL5574505 | — | — | 1 | 4.38 |
| CHEMBL5566343 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5570934 | — | IC50 | = | 8000.0 | nM | 5.10 |
| CHEMBL5555708 | — | IC50 | = | 8400.0 | nM | 5.08 |
| CHEMBL5572304 | — | IC50 | = | 11700.0 | nM | 4.93 |
| CHEMBL5570540 | — | IC50 | = | 13600.0 | nM | 4.87 |
| CHEMBL5573214 | — | IC50 | = | 14200.0 | nM | 4.85 |
| CHEMBL5569031 | — | IC50 | = | 15100.0 | nM | 4.82 |
| CHEMBL4297628 | RUXOTEMITIDE | IC50 | = | 16800.0 | nM | 4.78 |
| CHEMBL5569116 | — | IC50 | = | 18900.0 | nM | 4.72 |
| CHEMBL5592571 | — | IC50 | = | 36600.0 | nM | 4.44 |
| CHEMBL5574505 | — | IC50 | = | 41800.0 | nM | 4.38 |
| CHEMBL5566343 | — | IC50 | = | 210300.0 | nM | - |