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Assay Detail

CHEMBL5553500

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Anti-viral activity against RV-A 14 infected in human H1-HeLa cells incubated for 4 days by Cell Titer Glo assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Respiratory syncytial virus type A
Cell Type H1-HeLa
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Discovery of GS-7682, a Novel 4'-Cyano-Modified <i>C</i>-Nucleoside Prodrug with Broad Activity against Pneumo- and Picornaviruses and Efficacy in RSV-Infected African Green Monkeys.
Siegel DS, Hui HC, Pitts J, Vermillion MS, Ishida K, Rautiola D, Keeney M, Irshad H, Zhang L, Chun K, Chin G, Goyal B, Doerffler E, Yang H, Clarke MO, Palmiotti C, Vijjapurapu A, Riola NC, Stray K, Murakami E, Ma B, Wang T, Zhao X, Xu Y, Lee G, Marchand B, Seung M, Nayak A, Tomkinson A, Kadrichu N, Ellis S, Barauskas O, Feng JY, Perry JK, Perron M, Bilello JP, Kuehl PJ, Subramanian R, Cihlar T, Mackman RL.
J Med Chem (2024) 67 : 12945 -12968
PubMed 39018526 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 2 6.60 7.27

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5562532 1 7.27
CHEMBL1821850 1 5.92

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5562532 EC50 = 54.0 nM 7.27
CHEMBL1821850 EC50 = 1200.0 nM 5.92