Assay Detail
Functional
CHEMBL5576225
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Agonist activity at human GIPR expressed in CHO cells assessed as increase in cAMP production incubated for 30 mins by Eu-cAMP tracer based microplate reader analysis
25
Total Activities
25
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | CHO |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Gastric inhibitory polypeptide receptor (CHEMBL4383) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Design of a novel long-acting dual GLP-1/GIP receptor agonist.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 25 | 9.21 | 10.92 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5591096 | — | — | 1 | 10.92 |
| CHEMBL4297839 | TIRZEPATIDE | 4.0 | 1 | 10.52 |
| CHEMBL5591192 | — | — | 1 | 10.22 |
| CHEMBL5584064 | — | — | 1 | 10.19 |
| CHEMBL5584078 | — | — | 1 | 9.96 |
| CHEMBL5589666 | — | — | 1 | 9.85 |
| CHEMBL5595217 | — | — | 1 | 9.85 |
| CHEMBL5589598 | — | — | 1 | 9.70 |
| CHEMBL5589947 | — | — | 1 | 9.41 |
| CHEMBL5579723 | — | — | 1 | 9.38 |
| CHEMBL5593339 | — | — | 1 | 9.34 |
| CHEMBL5590213 | — | — | 1 | 9.22 |
| CHEMBL5593080 | — | — | 1 | 9.17 |
| CHEMBL5579773 | — | — | 1 | 9.14 |
| CHEMBL5595184 | — | — | 1 | 8.95 |
| CHEMBL5594125 | — | — | 1 | 8.88 |
| CHEMBL5589823 | — | — | 1 | 8.88 |
| CHEMBL5590197 | — | — | 1 | 8.73 |
| CHEMBL5590399 | — | — | 1 | 8.63 |
| CHEMBL5583949 | — | — | 1 | 8.59 |
| CHEMBL5593989 | — | — | 1 | 8.56 |
| CHEMBL5595154 | — | — | 1 | 8.43 |
| CHEMBL5591244 | — | — | 1 | 8.14 |
| CHEMBL5594494 | — | — | 1 | 7.83 |
| CHEMBL5595654 | — | — | 1 | 7.72 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5591096 | — | EC50 | = | 0.012 | nM | 10.92 |
| CHEMBL4297839 | TIRZEPATIDE | EC50 | = | 0.03 | nM | 10.52 |
| CHEMBL5591192 | — | EC50 | = | 0.06 | nM | 10.22 |
| CHEMBL5584064 | — | EC50 | = | 0.064 | nM | 10.19 |
| CHEMBL5584078 | — | EC50 | = | 0.11 | nM | 9.96 |
| CHEMBL5589666 | — | EC50 | = | 0.14 | nM | 9.85 |
| CHEMBL5595217 | — | EC50 | = | 0.14 | nM | 9.85 |
| CHEMBL5589598 | — | EC50 | = | 0.2 | nM | 9.70 |
| CHEMBL5589947 | — | EC50 | = | 0.39 | nM | 9.41 |
| CHEMBL5579723 | — | EC50 | = | 0.42 | nM | 9.38 |
| CHEMBL5593339 | — | EC50 | = | 0.46 | nM | 9.34 |
| CHEMBL5590213 | — | EC50 | = | 0.6 | nM | 9.22 |
| CHEMBL5593080 | — | EC50 | = | 0.67 | nM | 9.17 |
| CHEMBL5579773 | — | EC50 | = | 0.73 | nM | 9.14 |
| CHEMBL5595184 | — | EC50 | = | 1.12 | nM | 8.95 |
| CHEMBL5594125 | — | EC50 | = | 1.31 | nM | 8.88 |
| CHEMBL5589823 | — | EC50 | = | 1.31 | nM | 8.88 |
| CHEMBL5590197 | — | EC50 | = | 1.87 | nM | 8.73 |
| CHEMBL5590399 | — | EC50 | = | 2.33 | nM | 8.63 |
| CHEMBL5583949 | — | EC50 | = | 2.57 | nM | 8.59 |
| CHEMBL5593989 | — | EC50 | = | 2.76 | nM | 8.56 |
| CHEMBL5595154 | — | EC50 | = | 3.73 | nM | 8.43 |
| CHEMBL5591244 | — | EC50 | = | 7.2 | nM | 8.14 |
| CHEMBL5594494 | — | EC50 | = | 14.78 | nM | 7.83 |
| CHEMBL5595654 | — | EC50 | = | 19.19 | nM | 7.72 |