Assay Detail
Binding
CHEMBL5577680
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of human ALK1 using casein as substrate in presence of [gamma-33P]ATP and 10 uM ATP by radiometric assay
34
Total Activities
34
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Discovery of Two Highly Selective Structurally Orthogonal Chemical Probes for Activin Receptor-like Kinases 1 and 2.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 34 | 6.59 | 8.15 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4548795 | — | — | 1 | 8.15 |
| CHEMBL5083143 | — | — | 1 | 7.89 |
| CHEMBL5579725 | — | — | 1 | 7.60 |
| CHEMBL5590317 | — | — | 1 | 7.44 |
| CHEMBL5595157 | — | — | 1 | 7.39 |
| CHEMBL5592705 | — | — | 1 | 6.90 |
| CHEMBL5590255 | — | — | 1 | 6.87 |
| CHEMBL5593513 | — | — | 1 | 6.82 |
| CHEMBL5594766 | — | — | 1 | 6.44 |
| CHEMBL5590219 | — | — | 1 | 6.33 |
| CHEMBL5592288 | — | — | 1 | 6.30 |
| CHEMBL5592206 | — | — | 1 | 6.28 |
| CHEMBL5592629 | — | — | 1 | 6.09 |
| CHEMBL5594501 | — | — | 1 | 5.94 |
| CHEMBL5593369 | — | — | 1 | 5.88 |
| CHEMBL5593258 | — | — | 1 | 5.83 |
| CHEMBL5591254 | — | — | 1 | 5.69 |
| CHEMBL5590609 | — | — | 1 | 5.67 |
| CHEMBL5593123 | — | — | 1 | 5.66 |
| CHEMBL5589853 | — | — | 1 | - |
| CHEMBL5590714 | — | — | 1 | - |
| CHEMBL5594050 | — | — | 1 | - |
| CHEMBL5583693 | — | — | 1 | - |
| CHEMBL5591957 | — | — | 1 | - |
| CHEMBL5591016 | — | — | 1 | - |
| CHEMBL5595814 | — | — | 1 | - |
| CHEMBL5595327 | — | — | 1 | - |
| CHEMBL5595923 | — | — | 1 | - |
| CHEMBL5595818 | — | — | 1 | - |
| CHEMBL5594471 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4548795 | — | IC50 | = | 7.0 | nM | 8.15 |
| CHEMBL5083143 | — | IC50 | = | 13.0 | nM | 7.89 |
| CHEMBL5579725 | — | IC50 | = | 25.0 | nM | 7.60 |
| CHEMBL5590317 | — | IC50 | = | 36.0 | nM | 7.44 |
| CHEMBL5595157 | — | IC50 | = | 41.0 | nM | 7.39 |
| CHEMBL5592705 | — | IC50 | = | 125.0 | nM | 6.90 |
| CHEMBL5590255 | — | IC50 | = | 134.0 | nM | 6.87 |
| CHEMBL5593513 | — | IC50 | = | 152.0 | nM | 6.82 |
| CHEMBL5594766 | — | IC50 | = | 361.0 | nM | 6.44 |
| CHEMBL5590219 | — | IC50 | = | 466.0 | nM | 6.33 |
| CHEMBL5592288 | — | IC50 | = | 501.0 | nM | 6.30 |
| CHEMBL5592206 | — | IC50 | = | 524.0 | nM | 6.28 |
| CHEMBL5592629 | — | IC50 | = | 804.0 | nM | 6.09 |
| CHEMBL5594501 | — | IC50 | = | 1140.0 | nM | 5.94 |
| CHEMBL5593369 | — | IC50 | = | 1305.0 | nM | 5.88 |
| CHEMBL5593258 | — | IC50 | = | 1480.0 | nM | 5.83 |
| CHEMBL5591254 | — | IC50 | = | 2030.0 | nM | 5.69 |
| CHEMBL5590609 | — | IC50 | = | 2150.0 | nM | 5.67 |
| CHEMBL5593123 | — | IC50 | = | 2190.0 | nM | 5.66 |
| CHEMBL5589853 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL5590714 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL5594050 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL5583693 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL5591957 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL5591016 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL5595814 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL5595327 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL5595923 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL5595818 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL5594471 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL5591557 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL5595161 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL5583679 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL5595002 | — | IC50 | > | 3000.0 | nM | - |