Assay Detail
Binding
CHEMBL5577685
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of human ALK6 using casein as substrate in presence of [gamma-33P]ATP and 10 uM ATP by radiometric assay
34
Total Activities
34
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Bone morphogenetic protein receptor type-1B (CHEMBL5476) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Discovery of Two Highly Selective Structurally Orthogonal Chemical Probes for Activin Receptor-like Kinases 1 and 2.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 34 | 6.43 | 7.82 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5590317 | — | — | 1 | 7.82 |
| CHEMBL5083143 | — | — | 1 | 7.39 |
| CHEMBL4548795 | — | — | 1 | 7.06 |
| CHEMBL5595157 | — | — | 1 | 6.91 |
| CHEMBL5591254 | — | — | 1 | 6.28 |
| CHEMBL5594050 | — | — | 1 | 6.27 |
| CHEMBL5593513 | — | — | 1 | 6.27 |
| CHEMBL5590255 | — | — | 1 | 5.99 |
| CHEMBL5592705 | — | — | 1 | 5.95 |
| CHEMBL5592206 | — | — | 1 | 5.95 |
| CHEMBL5592629 | — | — | 1 | 5.94 |
| CHEMBL5595818 | — | — | 1 | 5.91 |
| CHEMBL5594766 | — | — | 1 | 5.86 |
| CHEMBL5583693 | — | — | 1 | - |
| CHEMBL5593258 | — | — | 1 | - |
| CHEMBL5589853 | — | — | 1 | - |
| CHEMBL5590714 | — | — | 1 | - |
| CHEMBL5592288 | — | — | 1 | - |
| CHEMBL5593369 | — | — | 1 | - |
| CHEMBL5591957 | — | — | 1 | - |
| CHEMBL5591016 | — | — | 1 | - |
| CHEMBL5595814 | — | — | 1 | - |
| CHEMBL5590219 | — | — | 1 | - |
| CHEMBL5579725 | — | — | 1 | - |
| CHEMBL5595923 | — | — | 1 | - |
| CHEMBL5591557 | — | — | 1 | - |
| CHEMBL5595161 | — | — | 1 | - |
| CHEMBL5583679 | — | — | 1 | - |
| CHEMBL5595002 | — | — | 1 | - |
| CHEMBL5590609 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5590317 | — | IC50 | = | 15.0 | nM | 7.82 |
| CHEMBL5083143 | — | IC50 | = | 41.0 | nM | 7.39 |
| CHEMBL4548795 | — | IC50 | = | 88.0 | nM | 7.06 |
| CHEMBL5595157 | — | IC50 | = | 123.0 | nM | 6.91 |
| CHEMBL5591254 | — | IC50 | = | 524.0 | nM | 6.28 |
| CHEMBL5594050 | — | IC50 | = | 536.0 | nM | 6.27 |
| CHEMBL5593513 | — | IC50 | = | 532.0 | nM | 6.27 |
| CHEMBL5590255 | — | IC50 | = | 1013.0 | nM | 5.99 |
| CHEMBL5592705 | — | IC50 | = | 1112.0 | nM | 5.95 |
| CHEMBL5592206 | — | IC50 | = | 1120.0 | nM | 5.95 |
| CHEMBL5592629 | — | IC50 | = | 1150.0 | nM | 5.94 |
| CHEMBL5595818 | — | IC50 | = | 1220.0 | nM | 5.91 |
| CHEMBL5594766 | — | IC50 | = | 1380.0 | nM | 5.86 |
| CHEMBL5594471 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL5594501 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL5595327 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL5593123 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL5583693 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL5593258 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL5589853 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL5590714 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL5592288 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL5593369 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL5591957 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL5591016 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL5595814 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL5590219 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL5579725 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL5595923 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL5591557 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL5595161 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL5583679 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL5595002 | — | IC50 | > | 3000.0 | nM | - |
| CHEMBL5590609 | — | IC50 | > | 3000.0 | nM | - |