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Assay Detail

CHEMBL5579423

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against Human parainfluenza virus 3 JS infected in human A549 cells assessed as reduction in viral proliferation incubated for 44 hrs by Hoechst dye based fluorescence analysis
7
Total Activities
7
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Human respirovirus 3
Confidence 1 — Organism
Curated By Autocuration

Target

Human respirovirus 3 (CHEMBL613126)
Type ORGANISM
Organism Human respirovirus 3

Publication

Discovery of Potent STT3A/B Inhibitors and Assessment of Their Multipathogen Antiviral Potential and Safety.
Pero JE, Mueller EA, Adams AM, Adolph RS, Bagchi P, Balce D, Bantscheff M, Barauskas O, Bartha I, Bohan D, Cai H, Carabajal E, Cassidy J, Cato M, Chaudhary KW, Chen D, Chen YP, Colas C, Darwech I, Eberl HC, Fernandez B, Gordon E, Grosse J, Hansen J, Hetzler B, Hwang S, Jeyasingh S, Kowalski B, Lehmann S, Lo G, McAllaster M, McHugh C, Momont C, Newby Z, Nigro M, Oladunni F, Pannirselvam M, Park A, Pearson N, Peat AJ, Plastridge B, Ranjan R, Safabakhsh P, Shapiro ND, Soriaga L, Stokes N, Sweeney D, Talecki L, Telenti A, Terrell A, Tse W, Wang L, Wang S, Wedel L, Werner T, Dalmas Wilk D, Yim S, Zhou J.
J Med Chem (2024) 67 : 14586 -14608
PubMed 39136957 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 7 7.43 8.22

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5595779 1 8.22
CHEMBL5583722 1 8.05
CHEMBL5583975 1 7.92
CHEMBL5583748 1 7.24
CHEMBL5591147 1 6.73
CHEMBL1720448 1 6.42
CHEMBL5589992 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5595779 EC50 = 6.0 nM 8.22
CHEMBL5583722 EC50 = 9.0 nM 8.05
CHEMBL5583975 EC50 = 12.0 nM 7.92
CHEMBL5583748 EC50 = 57.0 nM 7.24
CHEMBL5591147 EC50 = 187.0 nM 6.73
CHEMBL1720448 EC50 = 379.0 nM 6.42
CHEMBL5589992 EC50 - -