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Assay Detail

CHEMBL5581526

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antimalarial activity against Plasmodium falciparum W2 infected in RBC assessed as inhibition of growth incubated for 22 days by YOYO1 staining based LSR II flow cytometer
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Plasmodium falciparum
Cell Type RBC
Confidence 1 — Organism
Curated By Autocuration

Target

Plasmodium falciparum (CHEMBL364)
Type ORGANISM
Organism Plasmodium falciparum

Publication

Optimization of diastereomeric dihydropyridines as antimalarials.
Van Horn KS, Zhao Y, Parvatkar PT, Maier J, Mutka T, Lacrue A, Brockmeier F, Ebert D, Wu W, Casandra DR, Namelikonda N, Yacoub J, Sigal M, Knapp S, Floyd D, Waterson D, Burrows JN, Duffy J, DeRisi JL, Kyle DE, Guy RK, Manetsch R.
Eur J Med Chem (2024) 275 : 116599 -116599
PubMed 38909569 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 1 5.58 5.58

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL579338 1 5.58

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL579338 EC50 = 2613.0 nM 5.58