Assay Detail
Binding
CHEMBL5584805
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of COX-2 (unknown origin)
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Recent advances in c-Met-based dual inhibitors in the treatment of cancers.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.70 | 5.79 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5596467 | — | — | 1 | 5.79 |
| CHEMBL5596177 | — | — | 1 | 5.61 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5596467 | — | IC50 | = | 1620.0 | nM | 5.79 |
| CHEMBL5596177 | — | IC50 | = | 2430.0 | nM | 5.61 |