Assay Detail
Functional
CHEMBL5584935
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Cytotoxicity against human HeLa cells assessed as inhibition of cell growth incubated for 1 hr by MTT assay
30
Total Activities
30
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HeLa |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Rational design of a new short anticancer peptide with good potential for cancer treatment.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 30 | 5.07 | 6.03 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL412927 | MELITTIN | — | 1 | 6.03 |
| CHEMBL5591300 | — | — | 1 | 5.57 |
| CHEMBL5598040 | — | — | 1 | 5.54 |
| CHEMBL5589747 | — | — | 1 | 5.46 |
| CHEMBL5596081 | — | — | 1 | 5.41 |
| CHEMBL5597528 | — | — | 1 | 5.34 |
| CHEMBL5596674 | — | — | 1 | 5.33 |
| CHEMBL5598197 | — | — | 1 | 5.28 |
| CHEMBL5596119 | — | — | 1 | 5.26 |
| CHEMBL5596278 | — | — | 1 | 5.23 |
| CHEMBL5596860 | — | — | 1 | 5.15 |
| CHEMBL5598335 | — | — | 1 | 5.15 |
| CHEMBL5596777 | — | — | 1 | 5.12 |
| CHEMBL5598509 | — | — | 1 | 5.11 |
| CHEMBL5596841 | — | — | 1 | 5.09 |
| CHEMBL5596905 | — | — | 1 | 5.02 |
| CHEMBL5597709 | — | — | 1 | 4.92 |
| CHEMBL5598146 | — | — | 1 | 4.92 |
| CHEMBL5596501 | — | — | 1 | 4.89 |
| CHEMBL5598327 | — | — | 1 | 4.84 |
| CHEMBL5590181 | — | — | 1 | 4.83 |
| CHEMBL4297628 | RUXOTEMITIDE | 2.0 | 1 | 4.83 |
| CHEMBL5590137 | — | — | 1 | 4.79 |
| CHEMBL5597210 | — | — | 1 | 4.68 |
| CHEMBL5596132 | — | — | 1 | 4.65 |
| CHEMBL5598167 | — | — | 1 | 4.59 |
| CHEMBL5596207 | — | — | 1 | 4.49 |
| CHEMBL5596621 | — | — | 1 | 4.36 |
| CHEMBL5597409 | — | — | 1 | - |
| CHEMBL5596984 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL412927 | MELITTIN | IC50 | = | 934.0 | nM | 6.03 |
| CHEMBL5591300 | — | IC50 | = | 2676.0 | nM | 5.57 |
| CHEMBL5598040 | — | IC50 | = | 2873.0 | nM | 5.54 |
| CHEMBL5589747 | — | IC50 | = | 3453.0 | nM | 5.46 |
| CHEMBL5596081 | — | IC50 | = | 3938.0 | nM | 5.41 |
| CHEMBL5597528 | — | IC50 | = | 4537.0 | nM | 5.34 |
| CHEMBL5596674 | — | IC50 | = | 4628.0 | nM | 5.33 |
| CHEMBL5598197 | — | IC50 | = | 5225.0 | nM | 5.28 |
| CHEMBL5596119 | — | IC50 | = | 5525.0 | nM | 5.26 |
| CHEMBL5596278 | — | IC50 | = | 5908.0 | nM | 5.23 |
| CHEMBL5596860 | — | IC50 | = | 7153.0 | nM | 5.15 |
| CHEMBL5598335 | — | IC50 | = | 7046.0 | nM | 5.15 |
| CHEMBL5596777 | — | IC50 | = | 7588.0 | nM | 5.12 |
| CHEMBL5598509 | — | IC50 | = | 7852.0 | nM | 5.11 |
| CHEMBL5596841 | — | IC50 | = | 8142.0 | nM | 5.09 |
| CHEMBL5596905 | — | IC50 | = | 9456.0 | nM | 5.02 |
| CHEMBL5597709 | — | IC50 | = | 12050.0 | nM | 4.92 |
| CHEMBL5598146 | — | IC50 | = | 11920.0 | nM | 4.92 |
| CHEMBL5596501 | — | IC50 | = | 12920.0 | nM | 4.89 |
| CHEMBL5598327 | — | IC50 | = | 14360.0 | nM | 4.84 |
| CHEMBL5590181 | — | IC50 | = | 14660.0 | nM | 4.83 |
| CHEMBL4297628 | RUXOTEMITIDE | IC50 | = | 14700.0 | nM | 4.83 |
| CHEMBL5590137 | — | IC50 | = | 16330.0 | nM | 4.79 |
| CHEMBL5597210 | — | IC50 | = | 20770.0 | nM | 4.68 |
| CHEMBL5596132 | — | IC50 | = | 22160.0 | nM | 4.65 |
| CHEMBL5598167 | — | IC50 | = | 25840.0 | nM | 4.59 |
| CHEMBL5596207 | — | IC50 | = | 32190.0 | nM | 4.49 |
| CHEMBL5596621 | — | IC50 | = | 43720.0 | nM | 4.36 |
| CHEMBL5597409 | — | IC50 | = | 104200.0 | nM | - |
| CHEMBL5596984 | — | IC50 | = | 119700.0 | nM | - |