Assay Detail
Functional
CHEMBL5584938
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Cytotoxicity against human A549 cells assessed as inhibition of cell growth incubated for 1 hr by MTT assay
30
Total Activities
30
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | A549 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Rational design of a new short anticancer peptide with good potential for cancer treatment.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 30 | 4.94 | 5.74 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL412927 | MELITTIN | — | 1 | 5.74 |
| CHEMBL5596278 | — | — | 1 | 5.44 |
| CHEMBL5597528 | — | — | 1 | 5.43 |
| CHEMBL5596081 | — | — | 1 | 5.41 |
| CHEMBL5598040 | — | — | 1 | 5.41 |
| CHEMBL5591300 | — | — | 1 | 5.39 |
| CHEMBL5596119 | — | — | 1 | 5.30 |
| CHEMBL5589747 | — | — | 1 | 5.25 |
| CHEMBL5598197 | — | — | 1 | 5.22 |
| CHEMBL5596674 | — | — | 1 | 5.14 |
| CHEMBL5598335 | — | — | 1 | 5.09 |
| CHEMBL5598509 | — | — | 1 | 5.06 |
| CHEMBL5596841 | — | — | 1 | 5.04 |
| CHEMBL5596860 | — | — | 1 | 4.99 |
| CHEMBL5590181 | — | — | 1 | 4.96 |
| CHEMBL5596777 | — | — | 1 | 4.95 |
| CHEMBL5596905 | — | — | 1 | 4.84 |
| CHEMBL5590137 | — | — | 1 | 4.83 |
| CHEMBL5598146 | — | — | 1 | 4.81 |
| CHEMBL5598327 | — | — | 1 | 4.76 |
| CHEMBL5597709 | — | — | 1 | 4.73 |
| CHEMBL5596501 | — | — | 1 | 4.62 |
| CHEMBL5598167 | — | — | 1 | 4.31 |
| CHEMBL5597210 | — | — | 1 | 4.26 |
| CHEMBL4297628 | RUXOTEMITIDE | 2.0 | 1 | 4.19 |
| CHEMBL5596207 | — | — | 1 | 4.12 |
| CHEMBL5596621 | — | — | 1 | 4.06 |
| CHEMBL5596984 | — | — | 1 | - |
| CHEMBL5597409 | — | — | 1 | - |
| CHEMBL5596132 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL412927 | MELITTIN | IC50 | = | 1827.0 | nM | 5.74 |
| CHEMBL5596278 | — | IC50 | = | 3645.0 | nM | 5.44 |
| CHEMBL5597528 | — | IC50 | = | 3750.0 | nM | 5.43 |
| CHEMBL5596081 | — | IC50 | = | 3933.0 | nM | 5.41 |
| CHEMBL5598040 | — | IC50 | = | 3933.0 | nM | 5.41 |
| CHEMBL5591300 | — | IC50 | = | 4064.0 | nM | 5.39 |
| CHEMBL5596119 | — | IC50 | = | 5008.0 | nM | 5.30 |
| CHEMBL5589747 | — | IC50 | = | 5605.0 | nM | 5.25 |
| CHEMBL5598197 | — | IC50 | = | 5971.0 | nM | 5.22 |
| CHEMBL5596674 | — | IC50 | = | 7231.0 | nM | 5.14 |
| CHEMBL5598335 | — | IC50 | = | 8114.0 | nM | 5.09 |
| CHEMBL5598509 | — | IC50 | = | 8712.0 | nM | 5.06 |
| CHEMBL5596841 | — | IC50 | = | 9084.0 | nM | 5.04 |
| CHEMBL5596860 | — | IC50 | = | 10260.0 | nM | 4.99 |
| CHEMBL5590181 | — | IC50 | = | 10890.0 | nM | 4.96 |
| CHEMBL5596777 | — | IC50 | = | 11250.0 | nM | 4.95 |
| CHEMBL5596905 | — | IC50 | = | 14360.0 | nM | 4.84 |
| CHEMBL5590137 | — | IC50 | = | 14720.0 | nM | 4.83 |
| CHEMBL5598146 | — | IC50 | = | 15420.0 | nM | 4.81 |
| CHEMBL5598327 | — | IC50 | = | 17280.0 | nM | 4.76 |
| CHEMBL5597709 | — | IC50 | = | 18750.0 | nM | 4.73 |
| CHEMBL5596501 | — | IC50 | = | 23770.0 | nM | 4.62 |
| CHEMBL5598167 | — | IC50 | = | 49420.0 | nM | 4.31 |
| CHEMBL5597210 | — | IC50 | = | 55360.0 | nM | 4.26 |
| CHEMBL4297628 | RUXOTEMITIDE | IC50 | = | 64100.0 | nM | 4.19 |
| CHEMBL5596207 | — | IC50 | = | 75290.0 | nM | 4.12 |
| CHEMBL5596621 | — | IC50 | = | 87060.0 | nM | 4.06 |
| CHEMBL5596984 | — | IC50 | = | 482400.0 | nM | - |
| CHEMBL5597409 | — | IC50 | = | 530100.0 | nM | - |
| CHEMBL5596132 | — | IC50 | = | 131000.0 | nM | - |