Assay Detail
Functional
CHEMBL5585016
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antiproliferative activity against human CAL-51 cells assessed as inhibition of cell growth incubated for 72 hrs by MTT assay
17
Total Activities
17
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | CAL-51 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Hijacking monopolar spindle 1 (MPS1) for various cancer types by small molecular inhibitors: Deep insights from a decade of research and patents.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 17 | 7.31 | 8.10 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4086674 | — | — | 1 | 8.10 |
| CHEMBL4060730 | — | — | 1 | 8.05 |
| CHEMBL4068490 | — | — | 1 | 7.89 |
| CHEMBL4090966 | — | — | 1 | 7.82 |
| CHEMBL4086004 | — | — | 1 | 7.77 |
| CHEMBL4097084 | — | — | 1 | 7.75 |
| CHEMBL4063065 | — | — | 1 | 7.70 |
| CHEMBL4095765 | — | — | 1 | 7.52 |
| CHEMBL4066315 | — | — | 1 | 7.40 |
| CHEMBL4080975 | — | — | 1 | 7.22 |
| CHEMBL4062218 | — | — | 1 | 7.22 |
| CHEMBL4099734 | — | — | 1 | 7.16 |
| CHEMBL4065773 | — | — | 1 | 7.00 |
| CHEMBL4074116 | — | — | 1 | 6.92 |
| CHEMBL4063994 | — | — | 1 | 6.40 |
| CHEMBL4090356 | — | — | 1 | 6.30 |
| CHEMBL4064411 | — | — | 1 | 6.11 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4086674 | — | IC50 | = | 8.0 | nM | 8.10 |
| CHEMBL4060730 | — | IC50 | = | 9.0 | nM | 8.05 |
| CHEMBL4068490 | — | IC50 | = | 13.0 | nM | 7.89 |
| CHEMBL4090966 | — | IC50 | = | 15.0 | nM | 7.82 |
| CHEMBL4086004 | — | IC50 | = | 17.0 | nM | 7.77 |
| CHEMBL4097084 | — | IC50 | = | 18.0 | nM | 7.75 |
| CHEMBL4063065 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL4095765 | — | IC50 | = | 30.0 | nM | 7.52 |
| CHEMBL4066315 | — | IC50 | = | 40.0 | nM | 7.40 |
| CHEMBL4080975 | — | IC50 | = | 60.0 | nM | 7.22 |
| CHEMBL4062218 | — | IC50 | = | 60.0 | nM | 7.22 |
| CHEMBL4099734 | — | IC50 | = | 70.0 | nM | 7.16 |
| CHEMBL4065773 | — | IC50 | = | 100.0 | nM | 7.00 |
| CHEMBL4074116 | — | IC50 | = | 120.0 | nM | 6.92 |
| CHEMBL4063994 | — | IC50 | = | 400.0 | nM | 6.40 |
| CHEMBL4090356 | — | IC50 | = | 500.0 | nM | 6.30 |
| CHEMBL4064411 | — | IC50 | = | 770.0 | nM | 6.11 |