Assay Detail
Functional
CHEMBL5608633
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antagonist activity at CXCR4 (unknown origin) expressed in human HEK293FT cells
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HEK293FT |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Development and therapeutic perspectives of CXCR4 antagonists for disease therapy.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 1 | 9.52 | 9.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL237830 | — | — | 1 | 9.52 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL237830 | — | EC50 | = | 0.3 | nM | 9.52 |