Assay Detail
Functional
CHEMBL5608637
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Antagonist activity at CXCR4 (unknown origin) expressed in human HEK293T cells assessed as intracellular calcium flux by FLIPR assay
17
Total Activities
17
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HEK293T |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Development and therapeutic perspectives of CXCR4 antagonists for disease therapy.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 17 | 8.65 | 9.92 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5612607 | — | — | 1 | 9.92 |
| CHEMBL5612623 | — | — | 1 | 9.72 |
| CHEMBL5611972 | — | — | 1 | 9.72 |
| CHEMBL5613902 | — | — | 1 | 9.62 |
| CHEMBL4074140 | — | — | 1 | 9.00 |
| CHEMBL5614258 | — | — | 1 | 9.00 |
| CHEMBL5613857 | — | — | 1 | 9.00 |
| CHEMBL5613412 | — | — | 1 | 8.89 |
| CHEMBL4168957 | — | — | 1 | 8.68 |
| CHEMBL4162609 | — | — | 1 | 8.44 |
| CHEMBL1381819 | — | — | 1 | 8.42 |
| CHEMBL4172669 | — | — | 1 | 8.22 |
| CHEMBL4778921 | — | — | 1 | 8.06 |
| CHEMBL4075191 | — | — | 1 | 8.00 |
| CHEMBL5613701 | — | — | 1 | 7.62 |
| CHEMBL5612347 | — | — | 1 | 7.47 |
| CHEMBL4299893 | — | — | 1 | 7.27 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5612607 | — | EC50 | = | 0.12 | nM | 9.92 |
| CHEMBL5612623 | — | EC50 | = | 0.19 | nM | 9.72 |
| CHEMBL5611972 | — | EC50 | = | 0.19 | nM | 9.72 |
| CHEMBL5613902 | — | EC50 | = | 0.24 | nM | 9.62 |
| CHEMBL4074140 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL5614258 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL5613857 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL5613412 | — | EC50 | = | 1.3 | nM | 8.89 |
| CHEMBL4168957 | — | EC50 | = | 2.1 | nM | 8.68 |
| CHEMBL4162609 | — | EC50 | = | 3.6 | nM | 8.44 |
| CHEMBL1381819 | — | EC50 | = | 3.8 | nM | 8.42 |
| CHEMBL4172669 | — | EC50 | = | 6.0 | nM | 8.22 |
| CHEMBL4778921 | — | EC50 | = | 8.8 | nM | 8.06 |
| CHEMBL4075191 | — | EC50 | = | 10.0 | nM | 8.00 |
| CHEMBL5613701 | — | EC50 | = | 24.0 | nM | 7.62 |
| CHEMBL5612347 | — | EC50 | = | 34.0 | nM | 7.47 |
| CHEMBL4299893 | — | EC50 | = | 54.0 | nM | 7.27 |