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Assay Detail

CHEMBL5615281

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against Human rhinovirus 86 infected in human H1-HeLa cells assessed as reduction in cytopathic effect incubated for 72 hrs
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism rhinovirus B86
Cell Type H1-HeLa
Confidence 1 — Organism
Curated By Autocuration

Target

rhinovirus B86 (CHEMBL612480)
Type ORGANISM
Organism rhinovirus B86

Publication

7-Amino-3-phenyl-2-methyl-pyrazolopyrimidine derivatives inhibit human rhinovirus replication.
Chakrasali P, Hwang D, Lee JY, Jung E, Lee HL, Reneesh A, Skarka A, Musilek K, Nguyen NH, Shin JS, Jung YS.
Eur J Med Chem (2024) 276 : 116690 -116690
PubMed 39032404 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 3 7.38 8.22

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5618151 1 8.22
CHEMBL283403 ENVIROXIME 2.0 1 7.05
CHEMBL5619521 1 6.86

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5618151 EC50 = 6.0 nM 8.22
CHEMBL283403 ENVIROXIME EC50 = 89.0 nM 7.05
CHEMBL5619521 EC50 = 139.0 nM 6.86