Assay Detail
Binding
CHEMBL5620552
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of human recombinant PDE4
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 5 — Multiple protein complex / RNA |
| Curated By | Autocuration |
Publication
Advances in the development of phosphodiesterase 7 inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.81 | 5.85 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL182703 | — | — | 1 | 5.85 |
| CHEMBL183465 | — | — | 1 | 5.77 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL182703 | — | IC50 | = | 1420.0 | nM | 5.85 |
| CHEMBL183465 | — | IC50 | = | 1700.0 | nM | 5.77 |