Assay Detail
Binding
CHEMBL5621671
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Inhibition of TRPV1 (unknown origin)
6
Total Activities
6
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Transient receptor potential cation channel subfamily V member 1 (CHEMBL4794) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Transient receptor potential ankyrin 1 (TRPA1) modulators: Recent update and future perspective.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 6 | 5.04 | 5.06 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5558033 | — | — | 1 | 5.06 |
| CHEMBL511995 | LIQUIRITIN | — | 1 | 5.01 |
| CHEMBL1950590 | — | — | 1 | - |
| CHEMBL487732 | — | — | 1 | - |
| CHEMBL1950593 | — | — | 1 | - |
| CHEMBL1950595 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5558033 | — | IC50 | = | 8640.0 | nM | 5.06 |
| CHEMBL511995 | LIQUIRITIN | IC50 | = | 9800.0 | nM | 5.01 |
| CHEMBL1950590 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL487732 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1950593 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL1950595 | — | IC50 | > | 10000.0 | nM | - |